Pharmaceutical Chemistry

Drug Targets

Comprehensive drug target database including GPCRs, ion channels, nuclear receptors, kinases, and enzymes.

Drug Targets

Comprehensive drug target database including GPCRs, ion channels, nuclear receptors, kinases, and enzymes.

Browse the pages below for detailed information.

lysine demethylase 5D

lysine demethylase 5D — Enzyme drug target in the Histone demethylases family.

lysine demethylase 6A

lysine demethylase 6A — Enzyme drug target in the Histone demethylases family.

lysine demethylase 6B

lysine demethylase 6B — Enzyme drug target in the Histone demethylases family.

lysine demethylase 7A

lysine demethylase 7A — Enzyme drug target in the Histone demethylases family.

lysine demethylase 8

lysine demethylase 8 — Enzyme drug target in the Histone demethylases family.

lysine methyltransferase 2A

lysine methyltransferase 2A — Enzyme drug target in the Histone methyltransferases (HMTs) family.

lysine methyltransferase 2B

lysine methyltransferase 2B — Enzyme drug target in the Histone methyltransferases (HMTs) family.

lysine methyltransferase 2C

lysine methyltransferase 2C — Enzyme drug target in the Histone methyltransferases (HMTs) family.

lysine methyltransferase 2D

lysine methyltransferase 2D — Enzyme drug target in the Histone methyltransferases (HMTs) family.

lysine methyltransferase 2E (inactive)

lysine methyltransferase 2E (inactive) — Enzyme drug target in the Histone methyltransferases (HMTs) family.

lysine methyltransferase 5A

lysine methyltransferase 5A — Enzyme drug target in the Histone methyltransferases (HMTs) family.

lysine methyltransferase 5B

lysine methyltransferase 5B — Enzyme drug target in the Histone methyltransferases (HMTs) family.

lysine methyltransferase 5C

lysine methyltransferase 5C — Enzyme drug target in the Histone methyltransferases (HMTs) family.

lysophospholipase 1

lysophospholipase 1 — Enzyme drug target in the Hydrolases & Lipases family.

lysophospholipase 2

lysophospholipase 2 — Enzyme drug target in the Hydrolases & Lipases family.

lysyl oxidase

lysyl oxidase — Enzyme drug target in the Lysyl oxidases family.

lysyl oxidase like 2

lysyl oxidase like 2 — Enzyme drug target in the Lysyl oxidases family.

M1 receptor

M1 receptor — GPCR drug target in the Acetylcholine receptors (muscarinic) family.

M2 receptor

M2 receptor — GPCR drug target in the Acetylcholine receptors (muscarinic) family.

M3 receptor

M3 receptor — GPCR drug target in the Acetylcholine receptors (muscarinic) family.

M4 receptor

M4 receptor — GPCR drug target in the Acetylcholine receptors (muscarinic) family.

M5 receptor

M5 receptor — GPCR drug target in the Acetylcholine receptors (muscarinic) family.

magnesium transporter 1

magnesium transporter 1 — Transporter drug target in the SLC58 MagT-like magnesium transporter family family.

Major facilitator superfamily domain containing 7

Major facilitator superfamily domain containing 7 — Transporter drug target in the SLC49 family of FLVCR-related heme transporters family.

male germ cell associated kinase

male germ cell associated kinase — Enzyme drug target in the RCK family family.

Malonyl-CoA decarboxylase

Malonyl-CoA decarboxylase — Enzyme drug target in the Decarboxylases family.

MALT1 paracaspase

MALT1 paracaspase — Enzyme drug target in the C14: Caspase family.

maltase-glucoamylase

maltase-glucoamylase — Enzyme drug target in the Glycosidases family.

mannose-P-dolichol utilization defect 1

mannose-P-dolichol utilization defect 1 — Transporter drug target in the SLC66 Lysosomal amino acid transporters family.

MAPK activated protein kinase 2

MAPK activated protein kinase 2 — Enzyme drug target in the MAPKAPK subfamily family.

MAPK activated protein kinase 3

MAPK activated protein kinase 3 — Enzyme drug target in the MAPKAPK subfamily family.

MAPK activated protein kinase 5

MAPK activated protein kinase 5 — Enzyme drug target in the MAPKAPK subfamily family.

MAPK interacting serine/threonine kinase 1

MAPK interacting serine/threonine kinase 1 — Enzyme drug target in the MKN subfamily family.

MAPK interacting serine/threonine kinase 2

MAPK interacting serine/threonine kinase 2 — Enzyme drug target in the MKN subfamily family.

MAS1

MAS1 — GPCR drug target in the Mas1, BB3/Brs3, GPR17 family.

MAS1L

MAS1L — GPCR drug target in the Class A Orphans with emerging pharmacology family.

MATE2

MATE2 — Transporter drug target in the SLC47 family of multidrug and toxin extrusion transporters family.

maternal embryonic leucine zipper kinase

maternal embryonic leucine zipper kinase — Enzyme drug target in the MELK subfamily family.

MBL associated serine protease 2

MBL associated serine protease 2 — Enzyme drug target in the S1: Chymotrypsin family.

MC1 receptor

MC1 receptor — GPCR drug target in the Melanocortin receptors family.

MC2 receptor

MC2 receptor — GPCR drug target in the Melanocortin receptors family.

MC3 receptor

MC3 receptor — GPCR drug target in the Melanocortin receptors family.

MC4 receptor

MC4 receptor — GPCR drug target in the Melanocortin receptors family.

MC5 receptor

MC5 receptor — GPCR drug target in the Melanocortin receptors family.

MCH1 receptor

MCH1 receptor — GPCR drug target in the Melanin-concentrating hormone receptors family.

MCH2 receptor

MCH2 receptor — GPCR drug target in the Melanin-concentrating hormone receptors family.

MDM2 proto-oncogene

MDM2 proto-oncogene — Enzyme drug target in the E3 ubiquitin ligase components family.

mechanistic target of rapamycin kinase

mechanistic target of rapamycin kinase — Enzyme drug target in the FRAP subfamily family.

megakaryocyte-associated tyrosine kinase

megakaryocyte-associated tyrosine kinase — Enzyme drug target in the Csk family family.

membrane bound transcription factor peptidase, site 1

membrane bound transcription factor peptidase, site 1 — Enzyme drug target in the S8: Subtilisin family.

Membrane-associated transporter protein

Membrane-associated transporter protein — Transporter drug target in the SLC45 family of putative sugar transporters family.

methionine adenosyltransferase 2A

methionine adenosyltransferase 2A — Enzyme drug target in the Methionine turnover family.

Methionyl aminopeptidase 1

Methionyl aminopeptidase 1 — Enzyme drug target in the M24: Methionyl aminopeptidase family.

Methionyl aminopeptidase 2

Methionyl aminopeptidase 2 — Enzyme drug target in the M24: Methionyl aminopeptidase family.

Methionyl aminopeptidase type 1D (mitochondrial)

Methionyl aminopeptidase type 1D (mitochondrial) — Enzyme drug target in the M24: Methionyl aminopeptidase family.

methyltransferase 3, N6-adenosine-methyltransferase complex catalytic subunit

methyltransferase 3, N6-adenosine-methyltransferase complex catalytic subunit — Enzyme drug target in the Methyltransferases family.

mevalonate kinase

mevalonate kinase — Enzyme drug target in the Lanosterol biosynthesis pathway family.

MFSD2 lysolipid transporter A, lysophospholipid

MFSD2 lysolipid transporter A, lysophospholipid — Transporter drug target in the SLC59 Sodium-dependent lysophosphatidylcholine symporter family family.

MFSD2 lysolipid transporter B, sphingolipid

MFSD2 lysolipid transporter B, sphingolipid — Transporter drug target in the SLC59 Sodium-dependent lysophosphatidylcholine symporter family family.

MGC2541

MGC2541 — Transporter drug target in the SLC35 family of nucleotide sugar transporters family.